BIP! Finder - The war on hTG2: warhead optimization in small molecule human tissue transglutaminase inhibitors

2023 • The war on hTG2: warhead optimization in small molecule human tissue transglutaminase inhibitors

Authors: Lavleen Mader; Sarah K. I. Watt; Harish R. Iyer; Linh Nguyen; Harpreet Kaur; Jeffrey W. Keillor

Venue: RSC Medicinal Chemistry

Type: Publication

Abstract: This systematic structure–activity relationship study provides key insights into warhead design and application for optimizing efficiency, selectivity, and pharmacokinetic stability of hTG2 inhibitors.

Topics: Cell biology Biophysics Biochemistry

DOI: 10.1039/d2md00378c

BIP! social metrics: 0 45
External links: Crossref OpenAIRE

Related works: Dataset 1

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