2023 •
The war on hTG2: warhead optimization in small molecule human tissue transglutaminase inhibitors
Authors:
Lavleen Mader, Sarah K. I. Watt, Harish R. Iyer, Linh Nguyen, Harpreet Kaur, Jeffrey W. Keillor
Abstract:This systematic structure–activity relationship study provides key insights into warhead design and application for optimizing efficiency, selectivity, and pharmacokinetic stability of hTG2 inhibitors.
Lavleen Mader, Sarah K.I. Watt, Harish R. Iyer, Linh Nguyen, Harpreet Kaur, Jeffrey W Keillor
RSC Medicinal Chemistry ·
2022
 N/A
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