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2023 • The war on hTG2: warhead optimization in small molecule human tissue transglutaminase inhibitors

Authors: Lavleen Mader, Sarah K. I. Watt, Harish R. Iyer, Linh Nguyen, Harpreet Kaur, Jeffrey W. Keillor

Abstract: This systematic structure–activity relationship study provides key insights into warhead design and application for optimizing efficiency, selectivity, and pharmacokinetic stability of hTG2 inhibitors.

External links: OpenAIRE

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The War on hTG2: Warhead Optimization in Small Molecule Human Tissue Transglutaminase Inhi (...)

Lavleen Mader, Sarah K.I. Watt, Harish R. Iyer, Linh Nguyen, Harpreet Kaur, Jeffrey W Keillor

RSC Medicinal Chemistry · 2022

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